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Titolo Data di pubblicazione Autore(i) Rivista Editore
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function 2021 Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Ri...ta; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions 2021 Meleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira..., Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Mátyus, Péter; Maccioni, Elias MOLECULES
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives 2021 Meleddu, R.; Deplano, S.; Maccioni, E.; Ortuso, F.; Cottiglia, F.; Secci, D.; Onali, A.; Sanna, E....; Angeli, A.; Angius, R.; Alcaro, S.; Supuran, C. T.; Distinto, S. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Targeting HIV-1 RNase H: N'-(2-Hydroxy-benzylidene)-3,4,5-Trihydroxybenzoylhydrazone as Selective Inhibitor Active against NNRTIs-Resistant Variants 2020 Corona, Angela; Ballana, Ester; Distinto, Simona; Rogolino, Dominga; Del Vecchio, Claudia; Carcel...li, Mauro; Badia, Roger; Riveira-Muñoz, Eva; Esposito, Francesca; Parolin, Cristina; Esté, José A; Grandi, Nicole; Tramontano, Enzo VIRUSES
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation 2020 Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.;... Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII 2020 Meleddu, R.; Distinto, S.; Cottiglia, F.; Angius, R.; Caboni, P.; Angeli, A.; Melis, C.; Deplano,... S.; Alcaro, S.; Ortuso, F.; Supuran, C. T.; Maccioni, E. ACS MEDICINAL CHEMISTRY LETTERS
Quercetin blocks Ebola Virus infection by counteracting the VP24 Interferon inhibitory function 2020 Fanunza, Elisa; Iampietro, Mathieu; Distinto, Simona; Corona, Angela; Quartu, Marina; Maccioni, E...lias; Horvat, Branka; Tramontano, Enzo ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators 2019 Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Fi...lippo; Acquas, ELIO MARIA GIOACHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe JOURNAL OF NATURAL PRODUCTS
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids 2019 Meleddu, Rita; Petrikaite, Vilma; Distinto, Simona; Arridu, Antonella; Angius, Rossella; Serusi, ...Lorenzo; Škarnulytė, Laura; Endriulaitytė, Ugnė; Paškevičiu̅tė, Miglė; Cottiglia, Filippo; Gaspari, Marco; Taverna, Domenico; Deplano, Serenella; Fois, Benedetta; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases 2019 Distinto, S.; Meleddu, R.; Ortuso, F.; Cottiglia, F.; Deplano, S.; Sequeira, L.; Melis, C.; Fois,... B.; Angeli, A.; Capasso, C.; Angius, R.; Alcaro, S.; Supuran, C. T.; Maccioni, E. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Novel natural non-nucleoside inhibitors of HIV-1 reverse transcriptase identified by shape- and structure-based virtual screening techniques 2019 Costa, Giosuè; Rocca, Roberta; Corona, Angela; Grandi, Nicole; Moraca, Federica; Romeo, Isabella;... Talarico, Carmine; Giovanna Gagliardi, Maria; Alessandra Ambrosio, Francesca; Ortuso, Francesco; Alcaro, Stefano; Distinto, Simona; Maccioni, Elias; Tramontano, Enzo; Artese, Anna EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors 2019 Massari, Serena; Corona, Angela; Distinto, Simona; Desantis, Jenny; Caredda, Alessia; Sabatini, S...tefano; Manfroni, Giuseppe; Felicetti, Tommaso; Cecchetti, Violetta; Pannecouque, Christophe; Maccioni, Elias; Tramontano, Enzo; Tabarrini, Oriana JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors 2018 Melis, Claudia; Distinto, Simona; Bianco, Giulia; Meleddu, Rita; Cottiglia, Filippo; Fois, Benede...tta; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides 2018 Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Gaspari, Marco; Taverna, D...omenico; Melis, Claudia; Angeli, Andrea; Bianco, Giulia; Deplano, Serenella; Fois, Benedetta; Del Prete, Sonia; Capasso, Clemente; Alcaro, Stefano; Ortuso, Francesco; Yanez, Matilde; Supuran Claudiu, T.; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS
Identification of Myricetin as Ebolavirus VP35-dsRNA interaction inhibitor through a novel fluorescence-based assay 2018 Luca Daino, Gian; Frau, Aldo; Sanna, Cinzia; Rigano, Daniela; Distinto, Simona; Madau, Veronica; ...Esposito, Francesca; Fanunza, Elisa; Bianco, Giulia; Taglialatela-Scafati, Orazio; Zinzula, Luca; Maccioni, Elias; Corona, Angela; Tramontano, Enzo BIOCHEMISTRY
Identification of G-quadruplex DNA/RNA binders: Structure-based virtual screening and biophysical characterization 2017 Rocca, R.; Moraca, F.; Costa, G.; Nadai, M.; Scalabrin, M.; Talarico, C.; Distinto, S.; Maccioni,... E.; Ortuso, F.; Artese, A.; Alcaro, S.; Richter, S. N. BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase 2017 Sonar, Vijay P.; Corona, Angela; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Fois, Benedett...a; Floris, Costantino; Malpure, Nilesh V.; Alcaro, Stefano; Tramontano, Enzo; Cottiglia, Filippo EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors 2017 Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clement...e; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, Elias JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B 2017 Meleddu, Rita; Distinto, Simona; Cirilli, Roberto; Alcaro, Stefano; Yanez, Matilde; Sanna, Maria ...Luisa; Corona, Angela; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Maccioni, Elias JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase 2017 Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia...; Cottiglia, Filippo; Maccioni, Elias JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

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